1‐Substituted 2‐Azaspiro[3.3]heptanes: Overlooked Motifs for Drug Discovery

Angewchem
1‐Substituted 2‐Azaspiro[3.3]heptanes: Overlooked Motifs for Drug Discovery: The 2‐substituted piperidine core is found in drugs (18 FDA‐approved drugs), however, their spirocyclic analogues remain unknown. Described here is the synthesis of spirocyclic analogues for 2‐substituted...

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